Compile Data Set for Download or QSAR
Found 27 of ic50 data for polymerid = 50000507
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50259563(2-{[3,4-Dioxo-2-(pyridin-4-ylamino)cyclobut-1-en-1...)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of CK1-gamma1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7HK4PubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50259376(3-((R)-1-Phenyl-ethylamino)-4-(pyridin-4-ylamino)-...)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of CK1-gamma1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7HK4PubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50259532(2-{[3,4-Dioxo-2-(pyridin-4-ylamino)cyclobut-1-en-1...)copy SMILEScopy InChI
Affinity DataIC50: 520nMAssay Description:Inhibition of CK1-gamma1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7HK4PubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50259637(3-{[2-(2-Furyl)pyridin-4-yl]amino}-4-{[(1R)-1-phen...)copy SMILEScopy InChI
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of CK1-gamma1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7HK4PubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)copy SMILEScopy InChI
Affinity DataIC50: 5.52E+3nMAssay Description:Inhibition of CK1gamma1 (unknown origin) in presence of 5 mM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 7.17E+3nMAssay Description:Inhibition of human CK1gamma1 using KRRRAL[pS]VASLPGL as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5KB8PubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 7.44E+3nMAssay Description:Inhibition of human CK1gamma1 using KRRRAL[pS]VASLPGL as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W380MTPubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50311985(3-(7-(4-((1S,4S)-5-methyl-2,5-diazabicyclo[2.2.1]h...)copy SMILEScopy InChI
Affinity DataIC50: 9.51E+3nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z9510PubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50401152(CHEMBL2205766)copy SMILEScopy InChI
Affinity DataIC50: 9.55E+3nMAssay Description:Inhibition of CSNK1G1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ412BPubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50135286(CHEMBL3745885)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CK1gamma1 using [KRRRAL[pS]VASLPGL] as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7WT8PubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50519662(CHEMBL4438748)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human CK1gamma1(25 to 355 residues) using KRRRALS(p)VAS as substrate incubated for 40 mins in presence of [gamma-33ATP] by ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC93FGPubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50357884(CHEMBL1916359)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2HKRPubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50499634(CHEMBL3741589)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1gamma1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5CV4PubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50259638(3-{[2-(3-Thienyl)pyridin-4-yl]amino}-4-{[(1R)-1-ph...)copy SMILEScopy InChI
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of CK1-gamma1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7HK4PubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50316252(CHEMBL1095626 | methyl 4-(6-(4-aminophenyl)-4-morp...)copy SMILEScopy InChI
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3DGFPubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50094893(1-Amino-4-hydroxy-anthraquinone | 1-hydroxy-4-amin...)copy SMILEScopy InChI
Affinity DataIC50: 2.62E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7VGPPubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7VGPPubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50008516(IC261)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7VGPPubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50240382(1,4-Dihydroxyanthrachinon | 1,4-dihydroxy-9,10-ant...)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7VGPPubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50378568(CHEMBL1163016)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QJ7J72PubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315069(1-(4-(4-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-6-(t...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ08GKPubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50259601(3-{[2-(2-Fluorophenyl)pyridin-4-yl]amino}-4-{[(1R)...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CK1-gamma1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7HK4PubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50311954(6-methyl-4-(4-methyl-1H-indol-5-ylamino)-5-(3-(4-m...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD1Z1FPubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50311953(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(4-methylpipe...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD1Z1FPubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8T2GPubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50316253(CHEMBL1095627 | tert-Butyl 4-(6-(4-aminophenyl)-4-...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3DGFPubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human full-length GST-tagged CSNK1G1 expressed in baculovirus expression system using FRET-labeled Ser/Thr 05 peptide as su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed